| Bioactivity | ERK2 allosteric-IN-1 (compound 1) is a selective and allosteric ERK2 inhibitor with the IC50 of 11 μM[1]. |
| CAS | 872591-16-7 |
| Formula | C22H20N6O4 |
| Molar Mass | 432.43 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Sugiyama H, et al. Low entropic cost of binding confers high selectivity on an allosteric ERK2 inhibitor. Bioorg Med Chem Lett. 2023;93:129431. |