| Bioactivity | Dopamine D2 receptor agonist-3 (compound 3) is a selective D2 receptorpartial agonist and Dopamine D3 receptor antagonist (with pEC50 of 8.3 and <5.5 respectively)[1]. |
| In Vivo | Dopamine D2 receptor agonist-3 (3 mg/kg，皮下注射) 显示出较高的脑渗透性 (脑血比为 5.5) 和 Tmax 为 0.5 h[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
| CAS | 1257326-24-1 |
| Formula | C15H22ClN3O |
| Molar Mass | 295.81 |
| Appearance | 固体 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | 4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
| Reference | [1]. Holmes IP, et al. The identification of a selective dopamine D2 partial agonist, D3 antagonist displaying high levels of brain exposure. Bioorg Med Chem Lett. 2010 Mar 15;20(6):2013-6. |
Dopamine D2 receptor agonist-3
CAS: 1257326-24-1 F: C15H22ClN3O W: 295.81
Dopamine D2 receptor agonist-3 (compound 3) is a selective D2 receptorpartial agonist and Dopamine D3 receptor antagonis
Sales Email：peptidedb@qq.com
This product is for research use only, not for human use. We do not sell to patients.