| Bioactivity | Divaplon is a GABA receptor agonist with the EC50 values of 31 and 2 nM for α3β2γ2 and α5β2γ2, respectively. Divaplon shows non-sedating anxiolytic activity[1][2]. |
| CAS | 90808-12-1 |
| Formula | C17H17N3O2 |
| Molar Mass | 295.34 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Knoflach F, et al. Full and partial agonism displayed by benzodiazepine receptor ligands at recombinant gamma-aminobutyric acidA receptor subtypes. J Pharmacol Exp Ther. 1993;266(1):385-391. [2]. Sanger DJ, et al. Benzodiazepine (omega) receptor partial agonists and the acquisition of conditioned fear in mice. Psychopharmacology (Berl). 1995;121(1):104-108. |