| Bioactivity | D1R antagonist 1 (compound 12a) is a D1R antagonist, involved in G-protein- and β-arrestin-based signaling[1]. |
| Target | D1R |
| Name | D1R antagonist 1 |
| Formula | C22H26BrNO4 |
| Molar Mass | 448.35 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Namballa HK, et al. Discovery of Selective Dopamine Receptor Ligands Derived from (-)-Stepholidine via C-3 Alkoxylation and C-3/C-9 Dialkoxylation. J Med Chem. 2023 Jul 27;66(14):10060-10079. |