| Bioactivity | Cyclophilin inhibitor 1 is a potent and orally bioavailable cyclophilin A inhibitor, with a Kd of 5 nM, shows effective anti-HCV activity, with an EC50 of 98 nM for HCV 2a[1]. |
| Target | Kd: 5 nM (Cyclophilin A)EC50: 98 nM (HCV 2a) |
| Invitro | Cyclophilin inhibitor 1 (Compound 3) inhibits HCV 2a activity, with an EC50 of 98 nM[1]. |
| Name | Cyclophilin inhibitor 1 |
| CAS | 1509904-96-4 |
| Formula | C31H39N5O7 |
| Molar Mass | 593.67 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Mackman RL, et al. Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle. J Med Chem. 2018 Nov 8;61(21):9473-9499. |
Cyclophilin inhibitor 1
CAS: 1509904-96-4 F: C31H39N5O7 W: 593.67
Cyclophilin inhibitor 1 is a potent and orally bioavailable cyclophilin A inhibitor, with a Kd of 5 nM, shows effective
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