| Bioactivity | Cariprazine-d8 is a deuterium labeled Cariprazine. Cariprazine is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). |
| Name | Cariprazine-d8 |
| CAS | 1308278-50-3 |
| Formula | C21H24D8Cl2N4O |
| Molar Mass | 435.46 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Seneca N, et al. Occupancy of dopamine D2 and D3 and serotonin 5-HT1A receptors by the novel antipsychotic drug candidate, cariprazine (RGH-188), in monkey brain measured using positron emission tomography. Psychopharmacology (Berl). 2011 Dec;218(3):579-8 |
Cariprazine-d8
CAS: 1308278-50-3 F: C21H24D8Cl2N4O W: 435.46
Cariprazine-d8 is a deuterium labeled Cariprazine. Cariprazine is a novel antipsychotic drug candidate that exhibits hig
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