Bioactivity | CREBBP-IN-9 (Compound 9) is an inhibitor for CREBBP with an Kd of 29 μM[1]. |
CAS | 1219576-50-7 |
Formula | C16H15N5O2S |
Molar Mass | 341.39 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Xu M, et al., Discovery of CREBBP Bromodomain Inhibitors by High-Throughput Docking and Hit Optimization Guided by Molecular Dynamics. J Med Chem. 2016 Feb 25;59(4):1340-9. |