Bioactivity | CPN-267 (compound 7b) is a selective neuromedin U receptor 1 (NMUR1) agonist with the EC50 of 0.25 nM. CPN-267 suppresses body weight gain in mice and can be used for study of obesity[1]. |
CAS | 2241236-26-8 |
Sequence | {2-Thienylacetyl}-{Trp(α-Me}-Trp-Arg-Pro-Arg-Asn-NH2 |
Shortening | {2-Thienylacetyl}-{Trp(α-Me}-WRPRN-NH2 |
Formula | C50H66N16O8S |
Molar Mass | 1051.23 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Takayama K, et al. Discovery of a Human Neuromedin U Receptor 1-Selective Hexapeptide Agonist with Enhanced Serum Stability [published correction appears in J Med Chem. 2017 Sep 14;60(17):7613. |