| Bioactivity | CPI703, a BRD inhibitor, binds with residues in domain1 of 5DBM complex[1]. |
| Name | CPI703 |
| CAS | 1904649-00-8 |
| Formula | C17H22N4O |
| Molar Mass | 298.38 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Srimoyee Ghosh, et al. Regulatory T Cell Modulation by CBP/EP300 Bromodomain Inhibition. J Biol Chem. 2016 Jun 17;291(25):13014-27. [2]. Xue-Song Wang, et al. Theoretical research in structure characteristics of different inhibitors and differences of binding modes with CBP bromodomain. Bioorg Med Chem. 2018 Feb 1;26(3):712-720. |