| Bioactivity | CGP 56999 is a potent antagonist GABA(B) receptor, with the IC50 of 0.002 μM. CGP 56999 increased the levels of BDNF mRNA in the brain in vivo and in vitro[1]. |
| CAS | 153994-97-9 |
| Formula | C19H30NO5P |
| Molar Mass | 383.42 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. H. Bittiger, et al. GABAB Receptor Antagonists: Potential Therapeutic Applications. In: Tanaka, C., Bowery, N.G. (eds) GABA: Receptors, Transporters and Metabolism. Advances in Pharmacological Sciences. Birkhäuser Basel. |