| Bioactivity | BMS-986163 is a negative allosteric modulator of GluN2B. The prodrug BMS-986163 rapidly converts to its active parent molecule BMS-986169 (Ki=4 nM, IC50=24 nM). |
| Target | IC50: 24 nM (GluN2B, BMS-986169)Ki: 4 nM (GluN2B, BMS-986169) |
| Name | BMS-986163 |
| CAS | 1801151-09-6 |
| Formula | C23H28FN2O5P |
| Molar Mass | 462.45 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Marcin LR, et al. BMS-986163, a Negative Allosteric Modulator of GluN2B with Potential Utility in Major Depressive Disorder. ACS Med Chem Lett. 2018 Apr 13;9(5):472-477. |
BMS-986163
CAS: 1801151-09-6 F: C23H28FN2O5P W: 462.45
BMS-986163 is a negative allosteric modulator of GluN2B. The prodrug BMS-986163 rapidly converts to its active parent mo
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