| Bioactivity | Alverine citrate is a 5-HT1A receptor antagonist, with an IC50 of 101 nM. |
| Target | IC50: 101 nM (5-HT1A). |
| CAS | 150-59-4 |
| Formula | C20H27N |
| Molar Mass | 281.44 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Coelho, A.M., et al., Rectal antinociceptive properties of alverine citrate are linked to antagonism at the 5-HT1A receptor subtype. J Pharm Pharmacol, 2001. 53(10): p. 1419-26. [2]. Hayase, M., et al., Evolving mechanisms of action of alverine citrate on phasic smooth muscles. Br J Pharmacol, 2007. 152(8): p. 1228-38. |