Bioactivity | Ac-GpYLPQTV-NH2 is a STAT3 inhibitor with an IC50 value of 0.33 μM. Ac-GpYLPQTV-NH2 has antitumor activity[1]. |
Name | Ac-GpYLPQTV-NH2 |
CAS | 1349616-70-1 |
Sequence | Ac-Gly-{p-Tyr}-Leu-Pro-Gln-Thr-Val-NH2 |
Shortening | Ac-G-{p-Tyr}-LPQTV-NH2 |
Formula | C38H60N9O14P |
Molar Mass | 897.91 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Uehara Y, et al A. Novel high-throughput screening system for identifying STAT3-SH2 antagonists. Biochem Biophys Res Commun. 2009 Mar 13;380(3):627-31. |