| Bioactivity | AZ-PFKFB3-67 quarterhydrate is potent and selective metabolic kinase PFKFB3 inhibitor, with IC50s of 11, 159 and 1130 nM for PFKFB3, PFKFB2 and PFKFB1 respectively[1]. | ||||||||||||
| Target | IC50: 11 nM (PFKFB3), 159 nM (PFKFB2), 1130 nM (PFKFB1) | ||||||||||||
| Name | AZ-PFKFB3-67 quarterhydrate | ||||||||||||
| Formula | C26H25N5O3.1/4H2O | ||||||||||||
| Molar Mass | 460.01 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Boyd S, et al. Structure-Based Design of Potent and Selective Inhibitors of the Metabolic Kinase PFKFB3. J Med Chem. 2015;58(8):3611-3625. |
AZ-PFKFB3-67 quarterhydrate
CAS: F: C26H25N5O3.1/4H2O W: 460.01
AZ-PFKFB3-67 quarterhydrate is potent and selective metabolic kinase PFKFB3 inhibitor, with IC50s of 11, 159 and 1130 nM
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