| Bioactivity | AT1R antagonist 1 (compound 10) is a potent AT1R selective ligand. AT1R antagonist 1 exhibits a fair AT1R affinity, with a Ki of 8.5 nM[1]. |
| Target | Ki: 8.5 nM (AT1R), 320 nM (AT2R) |
| Name | AT1R antagonist 1 |
| Formula | C28H32F3N5O4S2 |
| Molar Mass | 623.71 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Bolteau R, et al. Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine. Eur J Med Chem. 2020 Mar 1;189:112078. |
AT1R antagonist 1
CAS: F: C28H32F3N5O4S2 W: 623.71
AT1R antagonist 1 (compound 10) is a potent AT1R selective ligand. AT1R antagonist 1 exhibits a fair AT1R affinity, with
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