| Bioactivity | A1AR antagonist 2 (compound 18h) is a potent A1 adenosine receptor (AR) antagonist with Kis of 1.49, 10.2, and 50.1 nM for hA1, hA2A and hA2B, respectively[1]. |
| Name | A1AR antagonist 2 |
| CAS | 1441961-74-5 |
| Formula | C17H12N4O |
| Molar Mass | 288.30 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Val C, et al. Optimization of 2-Amino-4,6-diarylpyrimidine-5-carbonitriles as Potent and Selective A1 Antagonists. J Med Chem. 2022;65(3):2091-2106. |
A1AR antagonist 2
CAS: 1441961-74-5 F: C17H12N4O W: 288.30
A1AR antagonist 2 (compound 18h) is a potent A1 adenosine receptor (AR) antagonist with Kis of 1.49, 10.2, and 50.1 nM f
Data collection：peptidedb@qq.com
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