Bioactivity | 4'-Raloxifene-β-D-glucopyranoside, a metabolite of Raloxifene, is a benzothiophene glucuronidated at the 4' postion. 4'-Raloxifene-β-D-glucopyranoside is a selective and orally active estrogen receptor antagonist. 4'-Raloxifene-β-D-glucopyranoside can be used for inhibiting bone loss and resorption, and lowering lipid levels. 4'-Raloxifene-β-D-glucopyranoside, example 5, is extracted from patent US5567820A[1]. |
Target | IC50: estrogen receptor |
Name | 4'-Raloxifene-β-D-glucopyranoside |
CAS | 334758-19-9 |
Formula | C34H37NO9S |
Molar Mass | 635.72 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Jeffrey A. Dodge, et al. Glucopyranoside benzothiophenes. Patent US5567820A. |