| Description | DEPTOR-IN-1 is an inhibitor of DEPTOR with a Kd of 9.3 μM. |
| Target activity | DEPTOR:9.3 μM (Kd) |
| molecular weight | 472.29 |
| Molecular formula | C24H16Cl2FNO4 |
| CAS | 2615911-12-9 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility | DMSO: 3.33 mg/mL (7.06 mM) |
| References | 1. Hou Y, et al. Design, Synthesis, and Biological Evaluation of Icaritin Derivatives as Novel Putative DEPTOR Inhibitors for Multiple Myeloma Treatment. J Med Chem. 2021 Oct 28;64(20):14942-14954. |