| Bioactivity | β2AR/M-receptor agonist-1 (example 131) is a muscarinic antagonist and β2 adrenoceptor agonist (MABA). β2AR/M-receptor agonist-1 shows potency to β2 adrenoceptor with an EC50 value of 9.2 nM. β2AR/M-receptor agonist-1 also has potency to muscarinic receptor with a Ki value of 30.2 nM. β2AR/M-receptor agonist-1 shows MABA potency with an EC50 value of 4.0 nM[1]. |
| In Vivo | β2AR/M-receptor agonist-1 (0.01 和 0.1 mg/kg；静脉注射，一次) 降低比格犬的心率[1]。 |
| Name | β2AR/M-receptor agonist-1 |
| CAS | 2230520-62-2 |
| Formula | C43H56BrN3O7 |
| Molar Mass | 806.82 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. WEN SHOUMING, et al. CLASS OF BIFUNCTIONAL COMPOUNDS WITH QUATERNARY AMMONIUM SALT STRUCTURE. WO2018108089. 2018. |
β2AR/M-receptor agonist-1
CAS: 2230520-62-2 F: C43H56BrN3O7 W: 806.82
β2AR/M-receptor agonist-1 (example 131) is a muscarinic antagonist and β2 adrenoceptor agonist (MABA). β2AR/M-recepto
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