Bioactivity | β2AR ligand 1 (Compound 4) is a homobivalent bitopic ligand for β2 adrenergic receptor (β2AR) on the orthosteric binding site (OBS) and the metastable binding sites (MBS)[1]. |
Formula | C33H49N5O4 |
Molar Mass | 579.77 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Gaiser BI, et al., Bitopic Ligands Support the Presence of a Metastable Binding Site at the β2 Adrenergic Receptor. J Med Chem. 2024 Jul 11;67(13):11053-11068. |