| Bioactivity | α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is a noncompetitive α-2,3-sialyltransferase inhibitor with an IC50 of 6 μM. | ||||||||||||
| Target | IC50: 6 μM (α-2,3-sialyltransferase) | ||||||||||||
| Invitro | α-2,3-sialyltransferase-IN-1 is compound 17 in the reference[1]. | ||||||||||||
| Name | α-2,3-sialyltransferase-IN-1 | ||||||||||||
| CAS | 881179-06-2 | ||||||||||||
| Formula | C28H45NO6 | ||||||||||||
| Molar Mass | 491.66 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
|
||||||||||||
| Reference | [1]. Chang KH, et al. Lithocholic acid analogues, new and potent alpha-2,3-sialyltransferase inhibitors. Chem Commun (Camb). 2006 Feb 14;(6):629-31. |