Bioactivity | α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is a noncompetitive α-2,3-sialyltransferase inhibitor with an IC50 of 6 μM. | ||||||||||||
Target | IC50: 6 μM (α-2,3-sialyltransferase) | ||||||||||||
Invitro | α-2,3-sialyltransferase-IN-1 is compound 17 in the reference[1]. | ||||||||||||
Name | α-2,3-sialyltransferase-IN-1 | ||||||||||||
CAS | 881179-06-2 | ||||||||||||
Formula | C28H45NO6 | ||||||||||||
Molar Mass | 491.66 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Chang KH, et al. Lithocholic acid analogues, new and potent alpha-2,3-sialyltransferase inhibitors. Chem Commun (Camb). 2006 Feb 14;(6):629-31. |