| Bioactivity | mPGES-1/sEH-IN-1 (compound 1f) is an inhibitor of sEH with IC50 value of 5 μM. mPGES-1/sEH-IN-1 shows antitumor activity with IC50 value of 25 µM via inhibts mPGES‐1[1]. |
| Formula | C20H16F3N3O2 |
| Molar Mass | 387.36 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Ester Colarusso, et al. 5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates. Arch Pharm (Weinheim). 2025 Jan;358(1):e2400708. |