| Bioactivity | hMcl-1-IN-1 (Compound 9) is an hMcl-1 inhibitor based on His224 aryl sulfonate fluoride, with an IC50 value of 5.8 nM[1]. |
| Target | IC50: 5.8 nM (hMcl-1). |
| Formula | C69H113FN20O19S |
| Molar Mass | 1577.82 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Alboreggia G, et al. Covalent Targeting of Histidine Residues with Aryl Fluorosulfates: Application to Mcl-1 BH3 Mimetics[J]. Journal of Medicinal Chemistry, 2024. |