| Bioactivity | hMCH-1R antagonist 1 (Compound 30) is an effective and selective antagonist of human melanin-concentrating hormone receptor 1 (hMCHR1) with an KB value of 3.6 nM. HMCH-1R antagonist 1 can bind to hMCHR1 and hMCHR2 with IC50 values of 65 nM and 49 nM, respectively. HMCH-1R antagonistist 1 can be used for metabolic research[1]. |
| Name | hMCH-1R antagonist 1 |
| CAS | 353487-64-6 |
| Sequence | Ac-Arg-Cys-Met-{5-Ava}-Arg-Val-Tyr-{5-Ava}-Cys-NH2 (Disulfide bridge: Cys2-Cys9) |
| Shortening | Ac-RCM-{5-Ava}-RVY-{5-Ava}-C-NH2 (Disulfide bridge: Cys2-Cys9) |
| Formula | C49H82N16O11S3 |
| Molar Mass | 1167.47 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
hMCH-1R antagonist 1
CAS: 353487-64-6 F: C49H82N16O11S3 W: 1167.47
hMCH-1R antagonist 1 (Compound 30) is an effective and selective antagonist of human melanin-concentrating hormone recep
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