Bioactivity | cBu-Cit-PROTAC BRD4 Degrader-5 is a cBu-Cit conjugated PROTAC degrader. cBu-Cit-PROTAC BRD4 Degrader-5 can potently degrade BRD4 in HER2 positive and negative breast cancer cell lines[1]. |
CAS | 2417369-73-2 |
Formula | C79H99ClN16O16S2 |
Molar Mass | 1628.31 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Marı A Maneiro, et al. Antibody-PROTAC Conjugates Enable HER2-Dependent Targeted Protein Degradation of BRD4. ACS Chem Biol. 2020 Jun 19;15(6):1306-1312. |