Bioactivity | c-Myc inhibitor 9 (compound 332) is a c-Myc inhibitor with an logEC50 of ≥6. c-Myc inhibitor 9 inhibits tumor growth in nude mouse models. c-Myc inhibitor 9 can be used for cancer research[1]. |
Invitro | c-Myc inhibitor 9 对 Myc 具有活性,在表达 c-Myc 的 A549 细胞中,logEC50 值 ≥6[1]。 |
In Vivo | c-Myc inhibitor 9 (3 mg/kg;腹腔注射,每周 2 次,49 天) 有效抑制 A549 异种移植裸鼠的肿瘤生长[1]。 Animal Model: |
Name | c-Myc inhibitor 9 |
CAS | 2799717-96-5 |
Formula | C27H31N5OS |
Molar Mass | 473.63 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Sheppard, David William, et al. Preparation of heteroaryl compounds as c-MYC mRNA translation modulators and uses thereof in the treatment of cancer. WO2022150316. 2022. |