| Bioactivity | Z8554052021 (compound 2021) is a potent CaSR and indeed GPCR positive allosteric modulator (PAM) with an EC50 of 3.3 nM. Z8554052021 has the potential for hyperparathyroidism research[1]. |
| Name | Z8554052021 |
| Formula | C21H21N3S |
| Molar Mass | 347.48 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Fangyu Liu, et al. Structure-based discovery of positive allosteric modulators for the calcium sensing receptor. bioRxiv,December 27, 2023. |