Bioactivity | YM471 free base is a non-peptide antagonist of vasopressin V1A and V2 receptors with potent and persistent antagonistic activity. YM471 exhibits high affinity for rat V1A and V2 receptors with K values of 0.16 and 0.77 nM, respectively[1]. |
CAS | 183173-00-4 |
Formula | C39H38F2N4O3 |
Molar Mass | 648.74 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Pharmacological characterization of YM471, a novel potent vasopressin V(1A) and V(2) receptor antagonist |