Bioactivity | Xanthoplanine, isolated from theroot of Xylopia parviflora, fully inhibits the EC50 ACh responses of both alpha7 and alpha4beta2 nACh receptors with estimated IC50 values of 9 μM (alpha7) and 5 μM (alpha4beta2)[1]. |
Name | Xanthoplanine |
CAS | 6872-88-4 |
Formula | C21H26NO4 |
Molar Mass | 356.43 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Iturriaga-Vásquez P, et al. Aporphine metho salts as neuronal nicotinic acetylcholine receptor blockers.Bioorg Med Chem. 2007 May 15;15(10):3368-72. |