| Bioactivity | Varenicline (Tartrate) (Standard) is the analytical standard of Varenicline (Tartrate). This product is intended for research and analytical applications. Varenicline (CP 526555) is an orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of α6β2 nAChR and a full agonist of α6β2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation. |
| CAS | 375815-87-5 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Varenicline Tartrate (Standard)
CAS: 375815-87-5 F: W:
Varenicline (Tartrate) (Standard) is the analytical standard of Varenicline (Tartrate). This product is intended for res
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This product is for research use only, not for human use. We do not sell to patients.