| Bioactivity | VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist that exhibits over a 10-fold increase in H3R binding affinity upon illumination at 360 nm. VUF14862 can be utilized for spatiotemporal studies of H3R signaling[1]. |
| CAS | 2223023-78-5 |
| Formula | C26H32N4O2 |
| Molar Mass | 432.56 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Hauwert NJ, et al. Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology. J Am Chem Soc. 2018 Mar 28;140(12):4232-4243. |
VUF14862
CAS: 2223023-78-5 F: C26H32N4O2 W: 432.56
VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist that exhibits over a 10-fold increase in H3R
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