| Bioactivity | VU6036864 (compound 45) is an orally active, selective mAChR M5 antagonist with IC50=20 nM for human M5. VU6036864 is >500-fold selective for human M1-4, with BBB characteristic and high oral bioavailability (%F>100%)[1]. |
| Target | IC50: 20 nM (human mAChR M5) |
| CAS | 2746406-36-8 |
| Formula | C15H12D4ClN5O3S |
| Molar Mass | 385.86 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Development of VU6036864: A Triazolopyridine-Based High-Quality Antagonist Tool Compound of the M5 Muscarinic Acetylcholine Receptor |
VU6036864
CAS: 2746406-36-8 F: C15H12D4ClN5O3S W: 385.86
VU6036864 (compound 45) is an orally active, selective mAChR M5 antagonist with IC50=20 nM for human M5. VU6036864 is >5
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