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VU6028418

CAS: 2649803-05-2 F: C23H27F3N4O W: 432.48

VU6028418 is a potent, highly selective and orally bioavailable M4 mAChR antagonist with an IC50 of 4.1 nM against hM4.
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Bioactivity VU6028418 is a potent, highly selective and orally bioavailable M4 mAChR antagonist with an IC50 of 4.1 nM against hM4[1].
In Vivo VU6028418 is orally bioavailable[1].In Vivo PK Parameters for VU6028418[1] parameter
Name VU6028418
CAS 2649803-05-2
Formula C23H27F3N4O
Molar Mass 432.48
Appearance Solid
Transport Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Reference [1]. Spock M, et al. Discovery of VU6028418: A Highly Selective and Orally Bioavailable M4 Muscarinic Acetylcholine Receptor Antagonist. ACS Med Chem Lett. 2021 Aug 2;12(8):1342-1349.

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Is for research use only, not for human use. We do not sell to patients.