Bioactivity | VDM11 is a potent and selective anandamide membrane transporter (AMT) inhibitor[1]. VDM11 inhibits FAAH and MAGL and may act as an alternative FAAH substrate[2]. |
CAS | 313998-81-1 |
Formula | C27H39NO2 |
Molar Mass | 409.60 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. De Petrocellis L, et al. Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin-like activity. FEBS Lett. 2000 Oct 13;483(1):52-6. [2]. Vandevoorde S, Fowler CJ. Inhibition of fatty acid amide hydrolase and monoacylglycerol lipase by the anandamide uptake inhibitor VDM11: evidence that VDM11 acts as an FAAH substrate. Br J Pharmacol. 2005 Aug;145(7):885-93. |