Bioactivity | UNC10099984A (Compound 6) is a functionally selective ligand for the dopamine D2 receptor, with a Ki value of 4.6 nM and an EC50 value of 6.2 nM for β-arrestin. UNC10099984A can be used for research into central nervous system disorders related to the D2 receptor[1]. |
Target | Ki:4.6 nM (D2).EC50: 6.2 nM (β-arrestin). |
CAS | 1354030-25-3 |
Formula | C24H29Cl2N3O2 |
Molar Mass | 462.41 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Jian Jin, et al. Functionally selective ligands of dopamine d2 receptors. Patent, WO2012003418, 2012-01-05. |