| Bioactivity | Tyropeptin A-4 (TP-101) is a potent proteasome inhibitor with the ability to inhibit mammalian 20S proteasome activity. Tyropeptin A-4 exerts its inhibitory effect by binding to the site responsible for trypsin-like activity. Tyropeptin A-4 derivative TP-104 has a 20-fold increase in inhibitory activity over Tyropeptin A. TP-110 specifically inhibits trypsin-like activity without affecting PGPH and trypsin-like activity[1]. |
| CAS | 688737-89-5 |
| Formula | C31H41N3O6 |
| Molar Mass | 551.67 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Structure-based design of derivatives of tyropeptin A as the potent and selective inhibitors of mammalian 20S proteasome |
Tyropeptin A-4
CAS: 688737-89-5 F: C31H41N3O6 W: 551.67
Tyropeptin A-4 (TP-101) is a potent proteasome inhibitor with the ability to inhibit mammalian 20S proteasome activity.
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