Bioactivity | Tianeptine metabolite MC5 sodium salt is a major active metabolite of tianeptine. Tianeptine and MC5 metabolite are eliminated with bile as glucuronide and glutamine conjugates[1]. |
In Vivo | Tianeptine 和 MC5 代谢物的平均消除半衰期分别为 1.16 和 7.53 小时[1]。 |
Name | Tianeptine metabolite MC5 sodium salt |
CAS | 115220-11-6 |
Formula | C19H20ClN2NaO4S |
Molar Mass | 430.88 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Szafarz M, et al. Pharmacokinetic study of tianeptine and its active metabolite MC5 in rats following different routes of administration using a novel liquid chromatography tandem mass spectrometry analytical method. Naunyn Schmiedebergs Arch Pharmacol. 2018 Feb;391(2):185-196. |