Bioactivity | Thalidomide-NH-amido-C4-Br is a conjugate of the E3 ligase ligand and the linker, that can be used for synthesis of PROTAC degrader BSJ-02-162 (HY-144995)[1]. |
CAS | 3027457-50-4 |
Formula | C19H21BrN4O5 |
Molar Mass | 465.30 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Nathanael S. Gray, et al. Degradation of cyclin-dependent kinase 4/6 (cdk4/6) by conjugation of cdk4/6 inhibitors with e3 ligase ligand and methods of use. WO2020023480 A1. |