| Bioactivity | TRPM8 antagonist 3 is a novel TRPM8 blocker with an IC50 value of 11 nM. | |||||||||
| Name | TRPM8 antagonist 3 | |||||||||
| CAS | 2102179-29-1 | |||||||||
| Formula | C13H12N2O4S | |||||||||
| Molar Mass | 292.31 | |||||||||
| Appearance | Solid | |||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | |||||||||
| Storage |
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| Reference | [1]. Bianchini G, et al. Discovery of Novel TRPM8 Blockers Suitable for the Treatment of Somatic and Ocular Painful Conditions: A Journey through pKa and LogD Modulation. J Med Chem. 2021 Nov 25;64(22):16820-16837. |