| Bioactivity | TP-680 is a cholecystokinin receptor antagonist. TP-680 binds 1510 times more strongly to rat pancreatic CCKA receptors (IC50=1.2 nM) than to rat brain CCKB receptors (IC50=1812.5 nM). TP-680 can be used in the study of gastrointestinal diseases[1]. |
| CAS | 176915-07-4 |
| Formula | C35H33N5O4S |
| Molar Mass | 619.73 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Akiyama T, et al. Pharmacological profile of TP-680, a new cholecystokininA receptor antagonist[J]. British journal of pharmacology, 1996, 117(7): 1558. |