| Bioactivity | TOP1288 is a narrow spectrum kinase inhibitor for P38α, Src and Syk kinase, with IC50 of 116nM, 24nM and 659nM, respectively. TOP1288 inhibits inflammatory cytokine release from inflamed biopsies and myofibroblasts[1]. |
| Target | IC50: 24 nM (Src), 116 nM (P38α), 659 nM (Syk) |
| CAS | 1630202-02-6 |
| Formula | C43H49N7O9S |
| Molar Mass | 839.96 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |