Bioactivity | TNKS1/2-IN-1 is a potent tankyrase TNKS1/2 inhibitor with pIC50s ranging from 7.1-8.2. TNKS1/2-IN-1 can be used for research of cancer, fibrosis, and other hyperproliferative diseases[1]. |
Target | TNKS1/2 |
Name | TNKS1/2-IN-1 |
CAS | 1498300-31-4 |
Formula | C26H23F4N3O4 |
Molar Mass | 517.47 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Keenan Richard M, et al. Preparation of quinazolinediones as tankyrase inhibitors for the treatment of cancer: World Intellectual Property Organization, WO2013177349 A2 2013-11-28. |