| Bioactivity | TGR5 agonist 5 (compound K91) is a potent agonist of TGR5, with EC50s of 19 μM and 30 μM in CRE-Luciferase assay anf cAMP accumulation assay, respectively[1]. |
| Formula | C22H26N2O2 |
| Molar Mass | 350.45 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. M Giovanna E Papadopoulos, et al. Discovery and characterization of small-molecule TGR5 ligands with agonistic activity. Eur J Med Chem. 2024 Jun 28:276:116616. |