| Bioactivity | TGR5 Receptor Agonist 4 is an agonist of Bile Acid Receptor (TGR5), with EC50 for hTGR5 and mTGR5 of 2 nM and 3 nM, respectively. TGR5 Receptor Agonist plays important roles in hypoglycemic and weight loss[1]. |
| Target | Bile Acid Receptor |
| Name | TGR5 Receptor Agonist 4 |
| CAS | 1872436-42-4 |
| Formula | C25H27ClN2O5 |
| Molar Mass | 470.95 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Sylvain Picon, et al. Discovery, Structure-Activity Relationships, and In Vivo Activity of Dihydropyridone Agonists of the Bile Acid Receptor TGR5. J Med Chem. 2023 Sep 14;66(17):11732-11760. |
TGR5 Receptor Agonist 4
CAS: 1872436-42-4 F: C25H27ClN2O5 W: 470.95
TGR5 Receptor Agonist 4 is an agonist of Bile Acid Receptor (TGR5), with EC50 for hTGR5 and mTGR5 of 2 nM and 3 nM, resp
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