Bioactivity | TC HSD 21 is a potent 17β-hydroxysteroid dehydrogenase type 3 (17β-HSD3) inhibitor with an IC50 of 14 nM. TC HSD 21 shows excellent selectivity over 17β-HSD isoenzymes and nuclear receptors[1]. | ||||||||||||
Target | IC50: 14 nM (17β-HSD3) | ||||||||||||
Name | TC HSD 21 | ||||||||||||
CAS | 330203-01-5 | ||||||||||||
Formula | C17H12BrNO3S2 | ||||||||||||
Molar Mass | 422.32 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Harada K,et al. Identification of oxazolidinediones and thiazolidinediones as potent 17β-hydroxysteroid dehydrogenase type 3 inhibitors. Bioorg Med Chem Lett. 2012 Jan 1;22(1):504-7. |