Bioactivity | TBK1/IKKε-IN-3 is a potent IP6K inhibitor with IC50 values of 3, 8.65 and 3.72 μM for IP6K1, IP6K2 and IP6K3, respectively. TBK1/IKKε-IN-3 can be used in the study of obesity diseases.[1]. |
Target | IC50: 3 μM (IP6K1), 8.65 μM (IP6K2), 3.72 μM (IP6K3) |
Name | TBK1/IKKε-IN-3 |
CAS | 851814-28-3 |
Formula | C16H11NO3 |
Molar Mass | 265.26 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Zhou Y, et al. Development of Novel IP6K Inhibitors for the Treatment of Obesity and Obesity-Induced Metabolic Dysfunctions. J Med Chem. 2022 May 12;65(9):6869-6887. |