PeptideDB

TASP0376377

CAS: 1233246-60-0 F: C25H16Cl2N2O4 W: 479.31

TASP0376377 is a potent and selective CRTH2 antagonist (IC50: 13 nM). TASP0376377 has binding affinity for CRTH2 (IC50:
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This product is for research use only, not for human use. We do not sell to patients.

Bioactivity TASP0376377 is a potent and selective CRTH2 antagonist (IC50: 13 nM). TASP0376377 has binding affinity for CRTH2 (IC50: 19 nM)[1].
Name TASP0376377
CAS 1233246-60-0
Formula C25H16Cl2N2O4
Molar Mass 479.31
Transport Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Reference [1]. Nishikawa-Shimono R, et al. Isoquinoline derivatives as potent CRTH2 antagonists: design, synthesis and SAR. Bioorg Med Chem. 2013 Dec 15;21(24):7674-85.