| Bioactivity | TAS2R14 agonist is a potent TAS2R14 partial agonist with an EC50 of 116.6 ±23.6 nM[1]. |
| Target | IC50: 116.6 nM (TAS2R14) |
| Invitro | 在 IP1 和 cAMP 积累试验中，TAS2R14 agonist 诱导 TAS2R14 激活，EC50 值分别为 100 nM 和 180 nM，与 IP1 和 cAMP 积累有关。 |
| Name | TAS2R14 agonist-1 |
| CAS | 2439115-08-7 |
| Formula | C15H9F6N5 |
| Molar Mass | 373.26 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Antonella Di Pizio, ret al. Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back. Cell Mol Life Sci. 2020 Feb;77(3):531-542. |