Bioactivity | TAAR1 agonist 2 (compound 30) is a full agonist of trace amine-associated receptor 1 (TAAR1) (pEC50=7.5). TAAR1 agonist 2 also exhibits agonist activity at H1 receptors and activates several members of the muscarinic acetylcholine receptor family, such as the M2 receptor (pEC50=5). TAAR1 agonist 2 can be used in the study of neuropsychiatric diseases[1]. |
CAS | 1804128-38-8 |
Formula | C9H11NO |
Molar Mass | 149.19 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Díaz-Holguín, et al. "AlphaFold accelerated discovery of psychotropic agonists targeting the trace amine–associated receptor 1." Science Advances 10.32 (2024): eadn1524. |