Bioactivity | T16A(inh)-C01 is an inhibitor of TMEM16A (ANO1). T16A(inh)-C01 blocks chloride channel mediated by ANO1 with an IC50 of 8.4 μM, without interfering with calcium signaling[1]. | ||||||||||||
Target | Target: Chloride Channel | ||||||||||||
Name | T16A(inh)-C01 | ||||||||||||
CAS | 171506-87-9 | ||||||||||||
Formula | C18H16O5 | ||||||||||||
Molar Mass | 312.32 | ||||||||||||
Appearance | Powder | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
|
||||||||||||
Reference | [1]. Namkung W, et al. TMEM16A inhibitors reveal TMEM16A as a minor component of calcium-activated chloride channel conductance in airway and intestinal epithelial cells. J Biol Chem. 2011 Jan 21. 286(3):2365-74. |